CHEBI ONTOLOGY - ANNOTATIONS
The Chemical Entities of Biological Interest (ChEBI) ontology is downloaded weekly from EMBL-EBI at http://www.ebi.ac.uk/chebi/ . The data is made available under the Creative Commons License (CC BY 3.0, http://creativecommons.org/licenses/by/3.0/ ). For more information see: Degtyarenko et al. (2008) ChEBI: a database and ontology for chemical entities of biological interest. Nucleic Acids Res. 36, D344–D350.
Term: EC 2.* (transferase) inhibitor
Accession: CHEBI:71300
browse the term
Definition: An enzyme inhibitor that inhibits the action of a transferase (EC 2.*)
Synonyms: related_synonym: EC 2 inhibitor; EC 2 inhibitors; EC 2.* (transferase) inhibitors; transferase inhibitor; transferase inhibitors
xref: Wikipedia:Transferase
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P2RY2
purinergic receptor P2Y2
multiple interactions
EXP
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acid inhibits the reaction [[Uridine Triphosphate results in increased activity of P2RY2 protein] which results in increased abundance of Arachidonic Acid]; pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acid inhibits the reaction [[Uridine Triphosphate results in increased activity of P2RY2 protein] which results in increased abundance of Cyclic AMP]
CTD
PMID:10604969
NCBI chr21:24,987,568...25,009,754
Ensembl chr21:24,992,848...24,996,059
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CLDN4
claudin 4
multiple interactions
EXP
pyrazolanthrone inhibits the reaction [Hydrogen Peroxide results in increased expression of CLDN4 protein]; pyrazolanthrone inhibits the reaction [Sodium Chloride results in increased expression of CLDN4 protein]
CTD
PMID:23816505
NCBI chr 6:6,492,706...6,506,750
Ensembl chr 6:6,493,513...6,494,145
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JUN
Jun proto-oncogene, AP-1 transcription factor subunit
multiple interactions
EXP
pyrazolanthrone inhibits the reaction [Sodium Chloride promotes the reaction [SP1 protein binds to JUN protein]]
CTD
PMID:23816505
NCBI chr 5:50,966,698...50,968,939
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MAPK8
mitogen-activated protein kinase 8
multiple interactions
EXP
pyrazolanthrone inhibits the reaction [Hydrogen Peroxide results in increased phosphorylation of MAPK8 protein]; pyrazolanthrone inhibits the reaction [Sodium Chloride results in increased phosphorylation of MAPK8 protein]
CTD
PMID:23816505
NCBI chr28:323,361...410,367
Ensembl chr28:368,513...406,401
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MAPK9
mitogen-activated protein kinase 9
multiple interactions
EXP
pyrazolanthrone inhibits the reaction [Hydrogen Peroxide results in increased phosphorylation of MAPK9 protein]; pyrazolanthrone inhibits the reaction [Sodium Chloride results in increased phosphorylation of MAPK9 protein]
CTD
PMID:23816505
NCBI chr11:1,443,528...1,480,501
Ensembl chr11:1,443,547...1,478,119
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SP1
Sp1 transcription factor
multiple interactions
EXP
pyrazolanthrone inhibits the reaction [Sodium Chloride promotes the reaction [SP1 protein binds to JUN protein]]; pyrazolanthrone inhibits the reaction [Sodium Chloride results in increased expression of SP1 protein]
CTD
PMID:23816505
NCBI chr27:1,802,587...1,861,187
Ensembl chr27:1,805,184...1,847,226
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CFTR
CF transmembrane conductance regulator
decreases activity
EXP
Genistein results in decreased activity of CFTR protein
CTD
PMID:15496164
NCBI chr14:56,290,417...56,452,919
Ensembl chr14:56,290,275...56,453,977
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CPNE6
copine 6
decreases activity
EXP
Genistein results in decreased activity of DHRS4 protein
CTD
PMID:17827741
NCBI chr 8:4,046,532...4,058,498
Ensembl chr 8:4,046,544...4,084,744
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CFTR
CF transmembrane conductance regulator
decreases activity
EXP
Glyburide results in decreased activity of CFTR protein
CTD
PMID:15496164
NCBI chr14:56,290,417...56,452,919
Ensembl chr14:56,290,275...56,453,977
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CCL17
C-C motif chemokine ligand 17
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL17 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] results in increased methylation of CCL17 promoter
CTD
PMID:33763461
NCBI chr 2:59,001,463...59,014,347
Ensembl chr 2:59,001,464...59,005,230
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CCL2
C-C motif chemokine ligand 2
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL2 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] results in increased methylation of CCL2 promoter
CTD
PMID:33763461
NCBI chr 9:39,008,187...39,009,932
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IL13
interleukin 13
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL17 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL2 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of IL31RA mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of TSLP mRNA]
CTD
PMID:33763461
NCBI chr11:20,957,870...20,961,391
Ensembl chr11:20,958,464...20,961,388
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IL31
interleukin 31
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL17 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL2 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of IL31RA mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of TSLP mRNA]
CTD
PMID:33763461
NCBI chr26:7,173,151...7,175,195
Ensembl chr26:7,172,451...7,175,195
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IL31RA
interleukin 31 receptor A
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of IL31RA mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] results in increased methylation of IL31RA promoter
CTD
PMID:33763461
NCBI chr 2:43,113,194...43,198,200
Ensembl chr 2:43,144,071...43,193,293
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IL4
interleukin 4
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL17 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of CCL2 mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of IL31RA mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of TSLP mRNA]
CTD
PMID:33763461
NCBI chr11:20,972,693...20,981,539
Ensembl chr11:20,972,690...20,981,534
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TSLP
thymic stromal lymphopoietin
multiple interactions
EXP
[Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] inhibits the reaction [[IL4 protein co-treated with IL13 protein co-treated with IL31 protein] results in increased expression of TSLP mRNA]; [Cannabidiol co-treated with Luteolin co-treated with 3,3',4,5'-tetrahydroxystilbene] results in increased methylation of TSLP promoter
CTD
PMID:33763461
NCBI chr 3:1,502,469...1,507,696
Ensembl chr 3:1,503,188...1,507,696
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PIK3CG
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma
multiple interactions
EXP
2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one inhibits the reaction [[Norepinephrine results in increased activity of PIK3CG protein] which results in increased chemical synthesis of phosphatidylinositol 3-phosphate]; 2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one inhibits the reaction [Norepinephrine results in increased activity of PIK3CG protein]
CTD
PMID:15958164
NCBI chr18:13,576,966...13,611,748
Ensembl chr18:13,570,999...13,611,141
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PRKCZ
protein kinase C zeta
multiple interactions
EXP
2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one inhibits the reaction [Clonidine results in increased phosphorylation of PRKCZ protein]; 2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one inhibits the reaction [Norepinephrine results in increased phosphorylation of PRKCZ protein]
CTD
PMID:15958164
NCBI chr 5:57,012,020...57,113,346
Ensembl chr 5:57,012,070...57,112,664
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ABCA5
ATP binding cassette subfamily A member 5
increases expression
EXP
masitinib results in increased expression of ABCA5 mRNA
CTD
PMID:22747577
NCBI chr 9:15,708,070...15,781,100
Ensembl chr 9:15,420,835...15,783,045
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ABHD14A
abhydrolase domain containing 14A
increases expression
EXP
masitinib results in increased expression of ABHD14A mRNA
CTD
PMID:22747577
NCBI chr20:37,738,500...37,744,689
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ABITRAM
actin binding transcription modulator
decreases expression
EXP
masitinib results in decreased expression of ABITRAM mRNA
CTD
PMID:22747577
NCBI chr11:64,094,653...64,100,078
Ensembl chr11:64,094,721...64,109,421
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ABLIM1
actin binding LIM protein 1
increases expression
EXP
masitinib results in increased expression of ABLIM1 mRNA
CTD
PMID:22747577
NCBI chr28:25,260,323...25,543,369
Ensembl chr28:25,260,873...25,545,304
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ACAT2
acetyl-CoA acetyltransferase 2
decreases expression
EXP
masitinib results in decreased expression of ACAT2 mRNA
CTD
PMID:22747577
NCBI chr 1:49,011,665...49,029,368
Ensembl chr 1:49,011,706...49,029,327
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ACSM3
acyl-CoA synthetase medium chain family member 3
increases expression
EXP
masitinib results in increased expression of ACSM3 mRNA
CTD
PMID:22747577
NCBI chr 6:24,558,010...24,594,326
Ensembl chr 6:24,558,142...24,582,728
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ACTL7A
actin like 7A
increases expression
EXP
masitinib results in increased expression of ACTL7A mRNA
CTD
PMID:22747577
NCBI chr11:64,031,305...64,033,908
Ensembl chr11:64,032,358...64,033,788
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ACTR2
actin related protein 2
decreases expression
EXP
masitinib results in decreased expression of ACTR2 protein
CTD
PMID:22747577
NCBI chr10:64,696,068...64,733,027
Ensembl chr10:64,696,111...64,730,553
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ADPRH
ADP-ribosylarginine hydrolase
increases expression
EXP
masitinib results in increased expression of ADPRH mRNA
CTD
PMID:22747577
NCBI chr33:23,218,633...23,226,844
Ensembl chr33:23,218,101...23,224,667
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AGA
aspartylglucosaminidase
increases expression
EXP
masitinib results in increased expression of AGA mRNA
CTD
PMID:22747577
NCBI chr16:52,314,860...52,324,879
Ensembl chr16:52,314,535...52,324,894
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AGO2
argonaute RISC catalytic component 2
decreases expression
EXP
masitinib results in decreased expression of AGO2 mRNA
CTD
PMID:22747577
NCBI chr13:35,169,243...35,230,252
Ensembl chr13:35,180,912...35,268,577
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AGRN
agrin
increases expression
EXP
masitinib results in increased expression of AGRN mRNA
CTD
PMID:22747577
NCBI chr 5:56,239,621...56,273,679
Ensembl chr 5:56,239,701...56,272,745
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AIG1
androgen induced 1
increases expression
EXP
masitinib results in increased expression of AIG1 mRNA
CTD
PMID:22747577
NCBI chr 1:34,643,994...34,884,445
Ensembl chr 1:34,643,764...34,884,119
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ALAS2
5'-aminolevulinate synthase 2
increases expression
EXP
masitinib results in increased expression of ALAS2 mRNA
CTD
PMID:22747577
NCBI chr X:46,703,477...46,731,767
Ensembl chr X:46,703,477...46,723,529
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ALDH5A1
aldehyde dehydrogenase 5 family member A1
decreases expression
EXP
masitinib results in decreased expression of ALDH5A1 mRNA
CTD
PMID:22747577
NCBI chr35:22,560,005...22,590,996
Ensembl chr35:22,560,008...22,587,875
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AMN1
antagonist of mitotic exit network 1 homolog
increases expression
EXP
masitinib results in increased expression of AMN1 mRNA
CTD
PMID:22747577
NCBI chr27:17,044,301...17,100,444
Ensembl chr27:17,044,309...17,361,570
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ANKRD26
ankyrin repeat domain containing 26
increases expression
EXP
masitinib results in increased expression of ANKRD26 mRNA
CTD
PMID:22747577
NCBI chr 2:6,230,466...6,402,360
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ANP32E
acidic nuclear phosphoprotein 32 family member E
decreases expression
EXP
masitinib results in decreased expression of ANP32E mRNA
CTD
PMID:22747577
NCBI chr17:59,460,864...59,482,467
Ensembl chr17:59,462,766...59,477,936
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ANXA1
annexin A1
increases expression
EXP
masitinib results in increased expression of ANXA1 protein
CTD
PMID:22747577
NCBI chr 1:84,744,159...84,763,011
Ensembl chr 1:84,744,163...84,763,011
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ANXA6
annexin A6
increases expression
EXP
masitinib results in increased expression of ANXA6 protein
CTD
PMID:22747577
NCBI chr 4:58,091,186...58,140,102
Ensembl chr 4:58,091,251...58,139,372
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ARMC12
armadillo repeat containing 12
increases expression
EXP
masitinib results in increased expression of ARMC12 mRNA
CTD
PMID:22747577
NCBI chr12:4,868,831...4,879,801
Ensembl chr12:4,869,774...4,879,793
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ASCC1
activating signal cointegrator 1 complex subunit 1
decreases expression
EXP
masitinib results in decreased expression of ASCC1 mRNA
CTD
PMID:22747577
NCBI chr 4:22,779,644...22,876,434
Ensembl chr 4:22,779,781...22,874,215
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B4GALT7
beta-1,4-galactosyltransferase 7
increases expression
EXP
masitinib results in increased expression of B4GALT7 mRNA
CTD
PMID:22747577
NCBI chr11:3,497,860...3,507,513
Ensembl chr11:3,498,153...3,505,034
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BIRC5
baculoviral IAP repeat containing 5
decreases expression
EXP
masitinib results in decreased expression of BIRC5 mRNA
CTD
PMID:22747577
NCBI chr 9:2,930,308...2,959,307
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BTBD3
BTB domain containing 3
decreases expression
EXP
masitinib results in decreased expression of BTBD3 mRNA
CTD
PMID:22747577
NCBI chr24:10,478,635...10,512,773
Ensembl chr24:10,479,900...10,512,185
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CA2
carbonic anhydrase 2
decreases expression
EXP
masitinib results in decreased expression of CA2 mRNA
CTD
PMID:22747577
NCBI chr29:31,959,225...31,975,309
Ensembl chr29:31,935,172...31,980,579
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CAMK2G
calcium/calmodulin dependent protein kinase II gamma
increases expression
EXP
masitinib results in increased expression of CAMK2G mRNA
CTD
PMID:22747577
NCBI chr 4:24,244,063...24,299,362
Ensembl chr 4:24,245,960...24,299,357
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CAPG
capping actin protein, gelsolin like
increases expression
EXP
masitinib results in increased expression of CAPG protein
CTD
PMID:22747577
NCBI chr17:39,619,429...39,640,944
Ensembl chr17:39,619,248...39,640,942
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CCT2
chaperonin containing TCP1 subunit 2
decreases expression
EXP
masitinib results in decreased expression of CCT2 protein
CTD
PMID:22747577
NCBI chr10:11,560,287...11,586,559
Ensembl chr10:11,560,396...11,578,433
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CD5L
CD5 molecule like
increases expression
EXP
masitinib results in increased expression of CD5L mRNA
CTD
PMID:22747577
NCBI chr 7:40,516,190...40,526,528
Ensembl chr 7:40,516,190...40,526,528
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CDADC1
cytidine and dCMP deaminase domain containing 1
increases expression
EXP
masitinib results in increased expression of CDADC1 mRNA
CTD
PMID:22747577
NCBI chr22:2,443,459...2,489,147
Ensembl chr22:2,436,206...2,489,016
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CDKN1A
cyclin dependent kinase inhibitor 1A
increases expression
EXP
masitinib results in increased expression of CDKN1A mRNA
CTD
PMID:22747577
NCBI chr12:5,746,898...5,755,103
Ensembl chr12:5,745,852...5,892,281
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CIAPIN1
cytokine induced apoptosis inhibitor 1
decreases expression
EXP
masitinib results in decreased expression of CIAPIN1 mRNA
CTD
PMID:22747577
NCBI chr 2:58,977,592...58,992,785
Ensembl chr 2:58,977,676...58,992,581
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CIRBP
cold inducible RNA binding protein
increases expression
EXP
masitinib results in increased expression of CIRBP mRNA
CTD
PMID:22747577
NCBI chr20:57,521,609...57,526,526
Ensembl chr20:57,519,119...57,526,435
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CLEC2B
C-type lectin domain family 2 member B
decreases expression
EXP
masitinib results in decreased expression of CLEC2B mRNA
CTD
PMID:22747577
NCBI chr27:36,088,754...36,143,581
Ensembl chr27:36,120,134...36,143,040
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CMTM7
CKLF like MARVEL transmembrane domain containing 7
increases expression
EXP
masitinib results in increased expression of CMTM7 mRNA
CTD
PMID:22747577
NCBI chr23:12,317,636...12,382,836
Ensembl chr23:12,328,303...12,382,837
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CORO1A
coronin 1A
increases expression
EXP
masitinib results in increased expression of CORO1A protein
CTD
PMID:22747577
NCBI chr 6:18,161,850...18,167,915
Ensembl chr 6:18,160,601...18,167,818
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CPNE1
copine 1
increases expression
EXP
masitinib results in increased expression of CPNE1 mRNA
CTD
PMID:22747577
NCBI chr24:24,554,636...24,589,748
Ensembl chr24:24,554,636...24,589,731
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CPNE6
copine 6
increases expression
EXP
masitinib results in increased expression of DHRS4 mRNA
CTD
PMID:22747577
NCBI chr 8:4,046,532...4,058,498
Ensembl chr 8:4,046,544...4,084,744
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CTSK
cathepsin K
increases expression
EXP
masitinib results in increased expression of CTSK mRNA
CTD
PMID:22747577
NCBI chr17:59,928,725...59,938,293
Ensembl chr17:59,929,287...59,938,507
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DLA-12
MHC class I DLA-12
increases expression
EXP
masitinib results in increased expression of DLA-12 mRNA
CTD
PMID:22747577
NCBI chr12:933,321...936,671
Ensembl chr12:932,613...987,561
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DLA-64
MHC class I DLA-64
increases expression
EXP
masitinib results in increased expression of DLA-64 mRNA
CTD
PMID:22747577
NCBI chr12:983,573...986,969
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DLGAP1
DLG associated protein 1
decreases expression
EXP
masitinib results in decreased expression of DLGAP1 mRNA
CTD
PMID:22747577
NCBI chr 7:70,082,563...70,949,116
Ensembl chr 7:70,081,885...70,406,213
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DLGAP5
DLG associated protein 5
decreases expression
EXP
masitinib results in decreased expression of DLGAP5 mRNA
CTD
PMID:22747577
NCBI chr 8:30,998,806...31,038,614
Ensembl chr 8:30,994,402...31,036,540
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DPCD
deleted in primary ciliary dyskinesia homolog
decreases expression
EXP
masitinib results in decreased expression of DPCD mRNA
CTD
PMID:22747577
NCBI chr28:14,201,302...14,219,121
Ensembl chr28:14,201,351...14,219,121
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DPYSL3
dihydropyrimidinase like 3
decreases expression
EXP
masitinib results in decreased expression of DPYSL3 mRNA
CTD
PMID:22747577
NCBI chr 2:41,687,725...41,809,402
Ensembl chr 2:41,690,845...41,802,376
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EBPL
EBP like
increases expression
EXP
masitinib results in increased expression of EBPL mRNA
CTD
PMID:22747577
NCBI chr22:2,116,588...2,137,935
Ensembl chr22:2,116,131...2,182,633
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EDEM2
ER degradation enhancing alpha-mannosidase like protein 2
increases expression
EXP
masitinib results in increased expression of EDEM2 mRNA
CTD
PMID:22747577
NCBI chr24:24,137,228...24,165,995
Ensembl chr24:24,137,228...24,165,968
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EIF3A
eukaryotic translation initiation factor 3 subunit A
decreases expression
EXP
masitinib results in decreased expression of EIF3A protein
CTD
PMID:22747577
NCBI chr28:29,290,668...29,326,851
Ensembl chr28:29,291,422...29,326,701
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EIF4A1
eukaryotic translation initiation factor 4A1
decreases expression
EXP
masitinib results in decreased expression of EIF4A1 protein
CTD
PMID:22747577
NCBI chr 5:32,495,606...32,500,805
Ensembl chr 5:32,484,572...32,500,805
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EIF5A2
eukaryotic translation initiation factor 5A2
decreases expression
EXP
masitinib results in decreased expression of EIF5A2 mRNA
CTD
PMID:22747577
NCBI chr34:35,309,812...35,322,382
Ensembl chr34:35,314,172...35,322,392
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ELSPBP1
epididymal sperm binding protein 1
increases expression
EXP
masitinib results in increased expression of ELSPBP1 mRNA
CTD
PMID:22747577
NCBI chr 1:108,159,609...108,187,224
Ensembl chr 1:108,159,611...108,188,076
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ETFDH
electron transfer flavoprotein dehydrogenase
decreases expression
EXP
masitinib results in decreased expression of ETFDH mRNA
CTD
PMID:22747577
NCBI chr15:55,752,170...55,781,118
Ensembl chr15:55,752,200...55,792,105
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GGT1
gamma-glutamyltransferase 1
increases expression
EXP
masitinib results in increased expression of GGT1 mRNA
CTD
PMID:22747577
NCBI chr26:28,301,455...28,315,029
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GKN1
gastrokine 1
increases expression
EXP
masitinib results in increased expression of GKN1 mRNA
CTD
PMID:22747577
NCBI chr10:67,788,329...67,793,445
Ensembl chr10:67,788,110...67,793,589
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GMFB
glia maturation factor beta
decreases expression
EXP
masitinib results in decreased expression of GMFB mRNA
CTD
PMID:22747577
NCBI chr 8:30,394,020...30,408,408
Ensembl chr 8:30,359,499...30,408,357
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GSTA4
glutathione S-transferase alpha 4
increases expression
EXP
masitinib results in increased expression of GSTA4 mRNA
CTD
PMID:22747577
NCBI chr12:20,426,724...20,443,200
Ensembl chr12:20,426,726...20,443,200
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GXYLT1
glucoside xylosyltransferase 1
decreases expression
EXP
masitinib results in decreased expression of GXYLT1 mRNA
CTD
PMID:22747577
NCBI chr27:11,754,609...11,810,245
Ensembl chr27:11,765,072...11,807,787
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HEBP2
heme binding protein 2
decreases expression
EXP
masitinib results in decreased expression of HEBP2 mRNA
CTD
PMID:22747577
NCBI chr 1:30,716,395...30,724,814
Ensembl chr 1:30,716,606...30,724,613
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HERPUD1
homocysteine inducible ER protein with ubiquitin like domain 1
increases expression
EXP
masitinib results in increased expression of HERPUD1 mRNA
CTD
PMID:22747577
NCBI chr 2:59,388,492...59,400,028
Ensembl chr 2:59,388,494...59,400,003
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HSP90B1
heat shock protein 90 beta family member 1
increases expression
EXP
masitinib results in increased expression of HSP90B1 protein
CTD
PMID:22747577
NCBI chr15:42,456,793...42,474,122
Ensembl chr15:42,456,764...42,579,311
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HTR2B
5-hydroxytryptamine receptor 2B
increases expression
EXP
masitinib results in increased expression of HTR2B mRNA
CTD
PMID:22747577
NCBI chr25:43,042,306...43,056,361
Ensembl chr25:43,042,173...43,056,612
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HYAL3
hyaluronidase 3
increases expression
EXP
masitinib results in increased expression of HYAL3 mRNA
CTD
PMID:22747577
NCBI chr20:39,041,940...39,047,388
Ensembl chr20:39,042,070...39,047,365
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IGFBP7
insulin like growth factor binding protein 7
increases expression
EXP
masitinib results in increased expression of IGFBP7 mRNA
CTD
PMID:22747577
NCBI chr13:49,138,406...49,207,235
Ensembl chr13:49,138,402...49,207,394
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IL13
interleukin 13
increases expression
EXP
masitinib results in increased expression of IL13 mRNA
CTD
PMID:22747577
NCBI chr11:20,957,870...20,961,391
Ensembl chr11:20,958,464...20,961,388
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IMMP2L
inner mitochondrial membrane peptidase subunit 2
increases expression
EXP
masitinib results in increased expression of IMMP2L mRNA
CTD
PMID:22747577
NCBI chr14:50,487,679...51,336,906
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IRX6
iroquois homeobox 6
increases expression
EXP
masitinib results in increased expression of IRX6 protein
CTD
PMID:22747577
NCBI chr 2:60,630,688...60,636,285
Ensembl chr 2:60,630,447...60,636,416
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ITGA6
integrin subunit alpha 6
decreases expression
EXP
masitinib results in decreased expression of ITGA6 mRNA
CTD
PMID:22747577
NCBI chr36:16,777,363...16,858,725
Ensembl chr36:16,776,863...16,855,449
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JAML
junction adhesion molecule like
decreases expression
EXP
masitinib results in decreased expression of JAML mRNA
CTD
PMID:22747577
NCBI chr 5:15,485,378...15,513,457
Ensembl chr 5:15,476,582...15,513,075
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JUN
Jun proto-oncogene, AP-1 transcription factor subunit
increases expression
EXP
masitinib results in increased expression of JUN mRNA
CTD
PMID:22747577
NCBI chr 5:50,966,698...50,968,939
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KCTD19
potassium channel tetramerization domain containing 19
increases expression
EXP
masitinib results in increased expression of KCTD19 mRNA
CTD
PMID:22747577
NCBI chr 5:82,060,946...82,093,248
Ensembl chr 5:82,061,449...82,093,246
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KLHL5
kelch like family member 5
increases expression
EXP
masitinib results in increased expression of KLHL5 mRNA
CTD
PMID:22747577
NCBI chr 3:73,258,925...73,347,262
Ensembl chr 3:73,262,895...73,344,879
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LBX2
ladybird homeobox 2
increases expression
EXP
masitinib results in increased expression of LBX2 mRNA
CTD
PMID:22747577
NCBI chr17:48,641,630...48,643,411
Ensembl chr17:48,641,674...48,643,239
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LIN7C
lin-7 homolog C, crumbs cell polarity complex component
decreases expression
EXP
masitinib results in decreased expression of LIN7C mRNA
CTD
PMID:22747577
NCBI chr21:48,061,446...48,071,458
Ensembl chr21:48,064,929...48,071,429
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LOC474850
heat shock 70 kDa protein 1-like
increases expression
EXP
masitinib results in increased expression of HSPA1L mRNA
CTD
PMID:22747577
NCBI chr12:1,281,164...1,285,010
Ensembl chr12:1,281,472...1,285,440
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LOC475707
GPN-loop GTPase 1
decreases expression
EXP
masitinib results in decreased expression of GPN1 mRNA
CTD
PMID:22747577
NCBI chr17:21,654,516...21,678,435
Ensembl chr17:21,545,673...21,673,157
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LOC478000
phytanoyl-CoA hydroxylase-like
increases expression
EXP
masitinib results in increased expression of PHYH mRNA
CTD
PMID:22747577
NCBI chr 2:23,185,901...23,206,719
Ensembl chr 2:23,185,782...23,253,497
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LOC609402
hemoglobin subunit beta-like
increases expression
EXP
masitinib results in increased expression of HBG1 mRNA
CTD
PMID:22747577
NCBI chr21:28,187,535...28,188,991
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LONRF1
LON peptidase N-terminal domain and ring finger 1
increases expression
EXP
masitinib results in increased expression of LONRF1 mRNA
CTD
PMID:22747577
NCBI chr16:36,220,324...36,256,896
Ensembl chr16:36,221,156...36,256,897
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LRP1
LDL receptor related protein 1
increases expression
EXP
masitinib results in increased expression of LRP1 mRNA
CTD
PMID:22747577
NCBI chr10:1,260,256...1,341,705
Ensembl chr10:1,260,719...1,352,271
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LRP8
LDL receptor related protein 8
decreases expression
EXP
masitinib results in decreased expression of LRP8 mRNA
CTD
PMID:22747577
NCBI chr 5:55,604,878...55,684,666
Ensembl chr 5:55,604,878...55,699,736
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LYRM1
LYR motif containing 1
increases expression
EXP
masitinib results in increased expression of LYRM1 mRNA
CTD
PMID:22747577
NCBI chr 6:24,428,461...24,460,291
Ensembl chr 6:24,441,307...24,460,331
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MAGEF1
MAGE family member F1
decreases expression
EXP
masitinib results in decreased expression of MAGEF1 mRNA
CTD
PMID:22747577
NCBI chr34:17,543,381...17,545,089
Ensembl chr34:17,543,906...17,544,868
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MOB1B
MOB kinase activator 1B
decreases expression
EXP
masitinib results in decreased expression of MOB1B mRNA
CTD
PMID:22747577
NCBI chr13:60,145,168...60,197,916
Ensembl chr13:60,145,366...60,195,463
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MPDZ
multiple PDZ domain crumbs cell polarity complex component
increases expression
EXP
masitinib results in increased expression of MPDZ mRNA
CTD
PMID:22747577
NCBI chr11:33,691,434...33,826,500
Ensembl chr11:33,692,296...33,826,437
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MYOZ1
myozenin 1
increases expression
EXP
masitinib results in increased expression of MYOZ1 mRNA
CTD
PMID:22747577
NCBI chr 4:24,158,532...24,165,416
Ensembl chr 4:24,158,720...24,165,392
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NAPG
NSF attachment protein gamma
decreases expression
EXP
masitinib results in decreased expression of NAPG mRNA
CTD
PMID:22747577
NCBI chr 7:76,403,561...76,424,994
Ensembl chr 7:76,403,595...76,423,170
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NDUFS1
NADH:ubiquinone oxidoreductase core subunit S1
decreases expression
EXP
masitinib results in decreased expression of NDUFS1 mRNA
CTD
PMID:22747577
NCBI chr37:14,680,908...14,713,838
Ensembl chr37:14,683,083...14,713,754
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NFKBIA
NFKB inhibitor alpha
increases expression
EXP
masitinib results in increased expression of NFKBIA mRNA
CTD
PMID:22747577
NCBI chr 8:14,100,203...14,103,453
Ensembl chr 8:14,100,671...14,103,433
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NRAS
NRAS proto-oncogene, GTPase
decreases expression
EXP
masitinib results in decreased expression of NRAS mRNA
CTD
PMID:22747577
NCBI chr17:52,411,733...52,418,788
Ensembl chr17:52,411,733...52,418,788
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NSG1
neuronal vesicle trafficking associated 1
decreases expression
EXP
masitinib results in decreased expression of NSG1 mRNA
CTD
PMID:22747577
NCBI chr 3:69,805,646...69,831,200
Ensembl chr 3:69,805,592...69,831,194
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NTRK1
neurotrophic receptor tyrosine kinase 1
increases expression
EXP
masitinib results in increased expression of NTRK1 mRNA
CTD
PMID:22747577
NCBI chr 7:41,140,931...41,159,326
Ensembl chr 7:41,140,879...41,159,288
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OCA2
OCA2 melanosomal transmembrane protein
decreases expression
EXP
masitinib results in decreased expression of OCA2 mRNA
CTD
PMID:22747577
NCBI chr 3:32,361,825...32,713,631
Ensembl chr 3:32,361,517...32,713,572
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OGT
O-linked N-acetylglucosamine (GlcNAc) transferase
increases expression
EXP
masitinib results in increased expression of OGT mRNA
CTD
PMID:22747577
NCBI chr X:55,821,227...55,857,597
Ensembl chr X:55,821,234...55,855,502
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OXCT1
3-oxoacid CoA-transferase 1
increases expression
EXP
masitinib results in increased expression of OXCT1 protein
CTD
PMID:22747577
NCBI chr 4:67,709,846...67,841,737
Ensembl chr 4:67,527,531...67,841,518
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PARP14
poly(ADP-ribose) polymerase family member 14
increases expression
EXP
masitinib results in increased expression of PARP14 mRNA
CTD
PMID:22747577
NCBI chr33:25,763,282...25,798,284
Ensembl chr33:25,763,255...25,798,198
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PCM1
pericentriolar material 1
increases expression
EXP
masitinib results in increased expression of PCM1 mRNA
CTD
PMID:22747577
NCBI chr16:41,212,733...41,291,654
Ensembl chr16:41,214,417...41,291,376
G
PCOLCE2
procollagen C-endopeptidase enhancer 2
decreases expression
EXP
masitinib results in decreased expression of PCOLCE2 mRNA
CTD
PMID:22747577
NCBI chr23:38,424,408...38,486,800
Ensembl chr23:38,426,216...38,487,252
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PDE6H
phosphodiesterase 6H
increases expression
EXP
masitinib results in increased expression of PDE6H mRNA
CTD
PMID:22747577
NCBI chr27:31,640,731...31,664,494
Ensembl chr27:31,640,737...31,664,401
G
PDHA1
pyruvate dehydrogenase E1 subunit alpha 1
decreases expression
EXP
masitinib results in decreased expression of PDHA1 mRNA
CTD
PMID:22747577
NCBI chr X:15,338,364...15,354,011
Ensembl chr X:15,338,202...15,387,458
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PDIA3
protein disulfide isomerase family A member 3
increases expression
EXP
masitinib results in increased expression of PDIA3 protein
CTD
PMID:22747577
NCBI chr30:10,487,926...10,513,437
Ensembl chr30:10,487,921...10,513,397
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PEBP4
phosphatidylethanolamine binding protein 4
increases expression
EXP
masitinib results in increased expression of PEBP4 mRNA
CTD
PMID:22747577
NCBI chr25:34,329,160...34,574,086
Ensembl chr25:34,317,421...34,574,066
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PECAM1
platelet and endothelial cell adhesion molecule 1
increases expression
EXP
masitinib results in increased expression of PECAM1 mRNA
CTD
PMID:22747577
NCBI chr 9:12,166,124...12,219,553
Ensembl chr 9:12,166,775...12,219,778
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PHF10
PHD finger protein 10
increases expression
EXP
masitinib results in increased expression of PHF10 mRNA
CTD
PMID:22747577
NCBI chr12:71,955,354...71,998,283
Ensembl chr12:71,787,082...71,998,243
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POMT1
protein O-mannosyltransferase 1
decreases expression
EXP
masitinib results in decreased expression of POMT1 mRNA
CTD
PMID:22747577
NCBI chr 9:52,615,349...52,631,538
Ensembl chr 9:52,615,655...52,630,836
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POR
cytochrome p450 oxidoreductase
increases expression
EXP
masitinib results in increased expression of POR mRNA
CTD
PMID:22747577
NCBI chr 6:7,247,780...7,316,282
Ensembl chr 6:7,263,574...7,316,297
G
PPA1
inorganic pyrophosphatase 1
decreases expression
EXP
masitinib results in decreased expression of PPA1 protein
CTD
PMID:22747577
NCBI chr 4:21,145,547...21,189,985
Ensembl chr 4:21,145,547...21,182,748
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PRPS2
phosphoribosyl pyrophosphate synthetase 2
decreases expression
EXP
masitinib results in decreased expression of PRPS2 mRNA
CTD
PMID:22747577
NCBI chr X:9,281,686...9,326,551
Ensembl chr X:9,281,730...9,418,289
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PSMB9
proteasome 20S subunit beta 9
increases expression
EXP
masitinib results in increased expression of PSMB9 mRNA
CTD
PMID:22747577
NCBI chr12:2,432,287...2,438,920
Ensembl chr12:2,432,505...2,438,069
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PSMD6
proteasome 26S subunit, non-ATPase 6
decreases expression
EXP
masitinib results in decreased expression of PSMD6 protein
CTD
PMID:22747577
NCBI chr20:27,206,801...27,220,059
G
PSMD9
proteasome 26S subunit, non-ATPase 9
decreases expression
EXP
masitinib results in decreased expression of PSMD9 mRNA
CTD
PMID:22747577
NCBI chr26:7,376,154...7,400,655
Ensembl chr26:7,377,413...7,400,573
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PTH
parathyroid hormone
increases expression
EXP
masitinib results in increased expression of PTH mRNA
CTD
PMID:22747577
NCBI chr21:36,417,062...36,419,967
Ensembl chr21:36,417,058...36,419,967
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PXYLP1
2-phosphoxylose phosphatase 1
decreases expression
EXP
masitinib results in decreased expression of ACPL2 mRNA
CTD
PMID:22747577
NCBI chr23:37,145,065...37,197,808
Ensembl chr23:37,145,086...37,196,427
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R3HDM2
R3H domain containing 2
increases expression
EXP
masitinib results in increased expression of R3HDM2 mRNA
CTD
PMID:22747577
NCBI chr10:1,377,664...1,504,008
Ensembl chr10:1,370,350...1,504,017
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RAB44
RAB44, member RAS oncogene family
increases expression
EXP
masitinib results in increased expression of RAB44 mRNA
CTD
PMID:22747577
NCBI chr12:5,769,056...5,804,963
Ensembl chr12:5,770,882...5,804,949
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RASGRP2
RAS guanyl releasing protein 2
increases expression
EXP
masitinib results in increased expression of RASGRP2 mRNA
CTD
PMID:22747577
NCBI chr18:52,412,331...52,426,910
Ensembl chr18:52,412,367...52,426,916
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RCAN1
regulator of calcineurin 1
increases expression
EXP
masitinib results in increased expression of RCAN1 mRNA
CTD
PMID:22747577
NCBI chr31:29,908,046...30,002,412
Ensembl chr31:29,909,388...30,002,418
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RGS13
regulator of G protein signaling 13
decreases expression
EXP
masitinib results in decreased expression of RGS13 mRNA
CTD
PMID:22747577
NCBI chr38:6,291,146...6,316,662
Ensembl chr38:6,291,182...6,315,198
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SAR1B
secretion associated Ras related GTPase 1B
decreases expression
EXP
masitinib results in decreased expression of SAR1A mRNA
CTD
PMID:22747577
NCBI chr11:22,713,459...22,743,190
Ensembl chr11:22,717,942...22,743,124
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SCD
stearoyl-CoA desaturase
decreases expression
EXP
masitinib results in decreased expression of SCD mRNA
CTD
PMID:22747577
NCBI chr28:13,112,741...13,129,129
Ensembl chr28:13,113,006...13,125,801
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SELENBP1
selenium binding protein 1
increases expression
EXP
masitinib results in increased expression of SELENBP1 protein
CTD
PMID:22747577
NCBI chr17:60,410,727...60,418,770
Ensembl chr17:60,410,734...60,418,704
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SERPINE2
serpin family E member 2
increases expression
EXP
masitinib results in increased expression of SERPINE2 mRNA
CTD
PMID:22747577
NCBI chr37:29,699,551...29,750,151
Ensembl chr37:29,700,024...29,724,228
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SFT2D2
SFT2 domain containing 2
decreases expression
EXP
masitinib results in decreased expression of SFT2D2 mRNA
CTD
PMID:22747577
NCBI chr 7:30,258,748...30,281,371
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SLA
Src like adaptor
increases expression
EXP
masitinib results in increased expression of SLA mRNA
CTD
PMID:22747577
NCBI chr13:29,503,304...29,590,679
Ensembl chr13:29,504,867...29,569,773
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SLC25A12
solute carrier family 25 member 12
decreases expression
EXP
masitinib results in decreased expression of SLC25A12 mRNA
CTD
PMID:22747577
NCBI chr36:16,185,011...16,391,080
Ensembl chr36:16,185,649...16,483,016
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SMC5
structural maintenance of chromosomes 5
decreases expression
EXP
masitinib results in decreased expression of SMC5 mRNA
CTD
PMID:22747577
NCBI chr 1:87,192,988...87,285,678
Ensembl chr 1:87,194,867...87,285,606
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SRR
serine racemase
increases expression
EXP
masitinib results in increased expression of SRR mRNA
CTD
PMID:22747577
G
STING1
stimulator of interferon response cGAMP interactor 1
increases expression
EXP
masitinib results in increased expression of TMEM173 mRNA
CTD
PMID:22747577
NCBI chr 2:34,783,947...34,792,204
Ensembl chr 2:34,784,232...34,789,072
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STOX1
storkhead box 1
increases expression
EXP
masitinib results in increased expression of STOX1 mRNA
CTD
PMID:22747577
NCBI chr 4:20,013,893...20,065,480
Ensembl chr 4:20,014,007...20,060,394
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STX16
syntaxin 16
increases expression
EXP
masitinib results in increased expression of STX16 mRNA
CTD
PMID:22747577
NCBI chr24:43,425,719...43,451,828
Ensembl chr24:43,426,470...43,449,077
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STYXL1
serine/threonine/tyrosine interacting like 1
increases expression
EXP
masitinib results in increased expression of STYXL1 mRNA
CTD
PMID:22747577
NCBI chr 6:7,323,911...7,389,878
Ensembl chr 6:7,316,477...7,389,842
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TARDBP
TAR DNA binding protein
decreases expression
EXP
masitinib results in decreased expression of TARDBP protein
CTD
PMID:22747577
NCBI chr 2:84,987,752...84,998,136
Ensembl chr 2:84,989,952...84,998,593
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TBC1D14
TBC1 domain family member 14
decreases expression
EXP
masitinib results in decreased expression of TBC1D14 mRNA
CTD
PMID:22747577
NCBI chr 3:58,992,743...59,097,581
Ensembl chr 3:58,926,237...59,097,621
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TCN2
transcobalamin 2
increases expression
EXP
masitinib results in increased expression of TCN2 mRNA
CTD
PMID:22747577
NCBI chr26:23,693,664...23,710,342
Ensembl chr26:23,693,773...23,709,832
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TCP1
t-complex 1
decreases expression
EXP
masitinib results in decreased expression of TCP1 protein
CTD
PMID:22747577
NCBI chr 1:49,029,260...49,038,023
Ensembl chr 1:49,029,282...49,038,020
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TEAD4
TEA domain transcription factor 4
increases expression
EXP
masitinib results in increased expression of TEAD4 mRNA
CTD
PMID:22747577
NCBI chr27:41,744,100...41,783,223
Ensembl chr27:41,748,871...41,803,556
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THEMIS2
thymocyte selection associated family member 2
decreases expression
EXP
masitinib results in decreased expression of THEMIS2 mRNA
CTD
PMID:22747577
NCBI chr 2:72,465,719...72,501,962
Ensembl chr 2:72,464,026...72,502,928
G
TM2D2
TM2 domain containing 2
increases expression
EXP
masitinib results in increased expression of TM2D2 mRNA
CTD
PMID:22747577
NCBI chr16:26,551,563...26,557,554
Ensembl chr16:26,551,628...26,556,285
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TMEM108
transmembrane protein 108
increases expression
EXP
masitinib results in increased expression of TMEM108 mRNA
CTD
PMID:22747577
NCBI chr23:29,992,038...30,331,791
Ensembl chr23:29,992,021...30,396,840
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TMEM260
transmembrane protein 260
increases expression
EXP
masitinib results in increased expression of TMEM260 mRNA
CTD
PMID:22747577
NCBI chr 8:32,238,992...32,309,320
Ensembl chr 8:32,238,988...32,306,317
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TNFSF10
TNF superfamily member 10
increases expression
EXP
masitinib results in increased expression of TNFSF10 mRNA
CTD
PMID:22747577
NCBI chr34:36,719,249...36,734,989
Ensembl chr34:36,670,849...36,735,060
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TNPO1
transportin 1
decreases expression
EXP
masitinib results in decreased expression of TNPO1 mRNA
CTD
PMID:22747577
NCBI chr 2:55,795,737...55,859,366
Ensembl chr 2:55,799,907...55,851,213
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TNS1
tensin 1
decreases expression
EXP
masitinib results in decreased expression of TNS1 mRNA
CTD
PMID:22747577
NCBI chr37:24,578,855...24,776,153
Ensembl chr37:24,581,806...24,808,049
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TOX
thymocyte selection associated high mobility group box
increases expression
EXP
masitinib results in increased expression of TOX mRNA
CTD
PMID:22747577
NCBI chr29:9,542,471...9,841,759
Ensembl chr29:9,544,561...9,842,034
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TSHB
thyroid stimulating hormone subunit beta
increases expression
EXP
masitinib results in increased expression of TSHB mRNA
CTD
PMID:22747577
NCBI chr17:52,659,137...52,685,388
Ensembl chr17:52,681,357...52,685,390
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TSPAN2
tetraspanin 2
increases expression
EXP
masitinib results in increased expression of TSPAN2 mRNA
CTD
PMID:22747577
NCBI chr17:52,692,744...52,749,048
Ensembl chr17:52,694,603...52,744,276
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TTC38
tetratricopeptide repeat domain 38
increases expression
EXP
masitinib results in increased expression of TTC38 protein
CTD
PMID:22747577
NCBI chr10:19,887,285...19,910,347
Ensembl chr10:19,773,373...19,910,683
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TTLL1
TTL family tubulin polyglutamylase complex subunit L1
decreases expression
EXP
masitinib results in decreased expression of TTLL1 mRNA
CTD
PMID:22747577
NCBI chr10:22,456,150...22,492,375
Ensembl chr10:22,456,146...22,488,505
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UCHL3
ubiquitin C-terminal hydrolase L3
increases expression
EXP
masitinib results in increased expression of UCHL3 protein
CTD
PMID:22747577
NCBI chr22:29,348,962...29,397,944
Ensembl chr22:29,348,706...29,407,965
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UQCC1
ubiquinol-cytochrome c reductase complex assembly factor 1
decreases expression
EXP
masitinib results in decreased expression of UQCC1 mRNA
CTD
PMID:22747577
NCBI chr24:24,285,147...24,381,819
Ensembl chr24:24,286,320...24,381,699
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UROD
uroporphyrinogen decarboxylase
increases expression
EXP
masitinib results in increased expression of UROD protein
CTD
PMID:22747577
NCBI chr15:15,313,808...15,317,130
Ensembl chr15:15,312,674...15,320,010
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UROS
uroporphyrinogen III synthase
increases expression
EXP
masitinib results in increased expression of UROS mRNA
CTD
PMID:22747577
NCBI chr28:34,952,074...34,983,532
Ensembl chr28:34,948,003...34,983,532
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VCPKMT
valosin containing protein lysine methyltransferase
decreases expression
EXP
masitinib results in decreased expression of VCPKMT mRNA
CTD
PMID:22747577
NCBI chr 8:26,611,333...26,636,700
Ensembl chr 8:26,625,677...26,636,316
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WAPL
WAPL cohesin release factor
decreases expression
EXP
masitinib results in decreased expression of WAPAL mRNA
CTD
PMID:22747577
NCBI chr 4:34,219,644...34,297,456
Ensembl chr 4:34,219,645...34,302,839
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YWHAZ
tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein zeta
increases expression
EXP
masitinib results in increased expression of YWHAZ protein
CTD
PMID:22747577
NCBI chr13:2,729,404...2,764,422
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ZNF23
zinc finger protein 23
increases expression
EXP
masitinib results in increased expression of ZNF23 mRNA
CTD
PMID:22747577
NCBI chr 5:77,246,374...77,260,761
Ensembl chr 5:77,246,667...77,260,350
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HEXB
hexosaminidase subunit beta
multiple interactions increases secretion
EXP
G(M1) Ganglioside inhibits the reaction [Melitten results in increased secretion of HEXB protein]; sialogangliosides inhibits the reaction [Melitten results in increased secretion of HEXB protein]; trisialoganglioside GT1 inhibits the reaction [Melitten results in increased secretion of HEXB protein]
CTD
PMID:21334356
NCBI chr 2:57,221,809...57,248,432
Ensembl chr 2:57,222,186...57,248,417
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ABCB1
ATP binding cassette subfamily B member 1
multiple interactions
EXP
[ML 7 results in decreased activity of MYLK protein] affects the reaction [ABCB1 protein affects the transport of Digoxin]
CTD
PMID:20510202
NCBI chr14:13,644,891...13,852,829
Ensembl chr14:13,542,647...13,742,727
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MYLK
myosin light chain kinase
multiple interactions
EXP
[ML 7 results in decreased activity of MYLK protein] affects the reaction [ABCB1 protein affects the transport of Digoxin]
CTD
PMID:20510202
NCBI chr33:26,663,991...26,867,370
Ensembl chr33:26,664,800...26,843,181
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IL6
interleukin 6
multiple interactions decreases expression
EXP
N-(2-(4-bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide inhibits the reaction [Amphotericin B results in increased expression of IL6 protein] N-(2-(4-bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide results in decreased expression of IL6 protein
CTD
PMID:24105867
NCBI chr14:36,474,268...36,478,519
Ensembl chr14:36,473,394...36,478,519
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PRKACB
protein kinase cAMP-activated catalytic subunit beta
multiple interactions
EXP
N-(2-(4-bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide inhibits the reaction [Amphotericin B results in increased expression of PRKACG protein]
CTD
PMID:24105867
NCBI chr 6:63,615,445...63,729,386
Ensembl chr 6:63,618,323...63,730,146
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PPARG
peroxisome proliferator activated receptor gamma
increases expression multiple interactions
EXP
Niacinamide results in increased expression of PPARG protein Resveratrol inhibits the reaction [Niacinamide results in increased expression of PPARG protein]
CTD
PMID:22539994
NCBI chr20:6,134,618...6,265,481
Ensembl chr20:6,050,357...6,207,981
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RUNX2
RUNX family transcription factor 2
increases acetylation multiple interactions decreases expression
EXP
Niacinamide results in increased acetylation of RUNX2 protein Niacinamide inhibits the reaction [SIRT1 protein binds to RUNX2 protein]; Resveratrol inhibits the reaction [Niacinamide inhibits the reaction [SIRT1 protein binds to RUNX2 protein]]; Resveratrol inhibits the reaction [Niacinamide results in decreased expression of RUNX2 protein]; Resveratrol inhibits the reaction [Niacinamide results in increased acetylation of RUNX2 protein]
CTD
PMID:22539994
NCBI chr12:13,723,535...13,842,565
Ensembl chr12:13,628,539...13,840,785 Ensembl chr12:13,628,539...13,840,785
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SIRT1
sirtuin 1
decreases expression multiple interactions
EXP
Niacinamide results in decreased expression of SIRT1 protein Niacinamide inhibits the reaction [SIRT1 protein binds to RUNX2 protein]; Resveratrol inhibits the reaction [Niacinamide inhibits the reaction [SIRT1 protein binds to RUNX2 protein]]; Resveratrol inhibits the reaction [Niacinamide results in decreased expression of SIRT1 protein]
CTD
PMID:22539994
NCBI chr 4:19,188,616...19,220,031
Ensembl chr 4:19,188,675...19,218,279
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REN
renin
decreases secretion multiple interactions
EXP
Ouabain results in decreased secretion of REN protein Vanadates inhibits the reaction [Ouabain results in decreased secretion of REN protein]
CTD
PMID:6093556
NCBI chr38:744,540...766,998
Ensembl chr38:744,614...755,012
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ABCB1
ATP binding cassette subfamily B member 1
multiple interactions
EXP
Quercetin inhibits the reaction [ABCB1 protein results in increased secretion of Ritonavir]
CTD
PMID:15266218
NCBI chr14:13,644,891...13,852,829
Ensembl chr14:13,542,647...13,742,727
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CPNE6
copine 6
decreases activity
EXP
Quercetin results in decreased activity of DHRS4 protein
CTD
PMID:17827741
NCBI chr 8:4,046,532...4,058,498
Ensembl chr 8:4,046,544...4,084,744
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HSP70
heat shock protein 70
decreases expression
EXP
Quercetin results in decreased expression of HSP70 protein
CTD
PMID:17009600
NCBI chr12:1,285,282...1,287,670
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ABCB1
ATP binding cassette subfamily B member 1
increases expression
EXP
Rifampin results in increased expression of ABCB1 mRNA; Rifampin results in increased expression of ABCB1 protein
CTD
PMID:22620706
NCBI chr14:13,644,891...13,852,829
Ensembl chr14:13,542,647...13,742,727
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NR1I2
nuclear receptor subfamily 1 group I member 2
increases activity
EXP
Rifampin results in increased activity of NR1I2 protein
CTD
PMID:27732639
NCBI chr33:23,444,367...23,456,405
Ensembl chr33:23,432,690...23,455,347
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CNR2
cannabinoid receptor 2
multiple interactions
EXP
SR 144528 binds to and results in decreased activity of CNR2 protein
CTD
PMID:21871882
NCBI chr 2:75,640,636...75,662,000
Ensembl chr 2:75,658,999...75,660,126
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PTGS2
prostaglandin-endoperoxide synthase 2
decreases expression
EXP
tolfenamic acid results in decreased expression of PTGS2 mRNA
CTD
PMID:15198222
NCBI chr 7:19,668,079...19,674,903
Ensembl chr 7:19,668,082...19,674,903
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HSP90B1
heat shock protein 90 beta family member 1
increases expression
EXP
Tunicamycin results in increased expression of HSP90B1 protein
CTD
PMID:17416481
NCBI chr15:42,456,793...42,474,122
Ensembl chr15:42,456,764...42,579,311
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HSPA5
heat shock protein family A (Hsp70) member 5
increases expression
EXP
Tunicamycin results in increased expression of HSPA5 protein
CTD
PMID:17416481
NCBI chr 9:57,850,870...57,855,607
Ensembl chr 9:57,850,922...57,855,257
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